Modular Click Chemistry Library: Searching for Better Functions

نویسندگان

چکیده

High throughput screening towards chemical libraries is the primary way to discover lead compounds in developing innovative drugs, especially new molecular entities. Accordingly, preparation of key step for drug development. Now, conventional small molecule and DNA-encoded are main models high-throughput screening. Recently, a model library, called modular click chemistry was proposed, which gives us an alternative choice construct high exhibits broad prospects accelerate Herein, this article mainly focuses on strategy prepare library.

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ژورنال

عنوان ژورنال: Chinese Journal of Chemistry

سال: 2021

ISSN: ['1614-7065', '1001-604X']

DOI: https://doi.org/10.1002/cjoc.202000596